Design of RGD-functionalized GSH-responsive pegylated polymeric protacs for selective BRD4 degradation and EndMT-driven cardiac fibrosis inhibition
设计RGD功能化的GSH响应性聚乙二醇化聚合物蛋白,用于选择性降解BRD4和抑制EndMT驱动的心脏纤维化
期刊:J Nanobiotechnology
影响因子:10.600
doi:10.1186/s12951-026-04036-7.
Tao Bi #,Lei Chen #,Ting Wang,Wenjun Miao,Silong Zhai,Rui Huang,Qin Sun,Yihan Chen,Hongna Su,Jie Zhou,Ruowen Li,Weixue Huang,Xiaojun Yao,Pei Luo,Zengjin Liu