Covalent Alkynylpyridopyrimidinones Targeting Cysteine 775 of the Epidermal Growth Factor Receptor Overcome Resistance to Current Therapies
共价炔基吡啶并嘧啶酮靶向表皮生长因子受体的半胱氨酸775,克服对现有疗法的耐药性
期刊:J Med Chem
影响因子:6.800
doi:10.1021/acs.jmedchem.5c02924
Hannah L Stewart,Cinzia Bordoni,Claire E Jennings,Islam Al-Khawaldeh,Mathew P Martin,Richard A Noble,Nicole Phillips,Sara Pintar,Lisa Prendergast,Huw D Thomas,Lan-Z Wang,Jessica E Watt,Anita Wittner,Agnieszka K Bronowska,Céline Cano,Martin E M Noble,Stephen R Wedge,Michael J Waring